GW842166X

  • Chemical Properties
CAS No. 666260-75-9 Cat. No. BCP05306
Name GW842166X
Synonyms GW 842166X;GW-842166X;
Formula C18H17Cl2F3N4O2 M. Wt 449.26
  • Biological Activity
Description GW842166X shows similar potency and efficacy for rat and human recombinant CB2 receptors with EC50 of 91 nM and 63nM, respectively.GW-842166X exhibits full agonist potency with an EC50 of 133 nM and Emax of 101% in cyclase assays. GW-842166X exhibits weak agonist potency with an EC50 of 7.780 μM and Emax of 84% in FLIPR assays.
Pathways GPCR/G Protein 
Targets Cannabinoid Receptor 

Structure

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