马罗匹坦
CAS号 | 147116-67-4 | 货号 | BCP29857 |
中文名 | 马罗匹坦 | ||
英文名 | Maropitant | ||
中文别名 | |||
英文别名 | CJ-11,972; CJ 11,972; CJ11,972; CJ-11972; CJ 11972; CJ11972; | ||
分子式 | C32H40N2O | 分子量 | 468.67 |
生物活性 | Maropitan, also known as CJ 11972, is a neurokinin (NK1) receptor antagonist, which was developed by Zoetis specifically for the treatment of motion sickness and vomiting in dogs. It was approved by the FDA in 2007 for use in dogs, and more recently has also been approved for use in cats. | ||
信号通路 | GPCR/G Protein | ||
靶 点 | NK Receptor |
结构式

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