Rimegepant sulfate hydrate

  • Chemical Properties
CAS No. 1374024-48-2 Cat. No. BCP42168
Name Rimegepant sulfate hydrate
Synonyms Rimegepant sulfate;BHV-3000; BHV 3000; BHV3000; BMS-927711; BMS 927711; BMS927711;
Formula C56H64F4N12O13S M. Wt 1221.25
  • Biological Activity
Description Rimegepant is a potent, selective, competitive, and orally active calcitonin gene-related peptide (CGRP) antagonist in clinical trials for treating migraines. Rimegepant has shown in vivo efficacy without vasoconstriction effect. BMS-927711 is superior to placebo at several different doses (75 mg, 150 mg, and 300 mg) and has an excellent tolerability profile.
Pathways Neuro Signaling Pathway GPCR/G Protein 
Targets CGRP Receptor 

Structure

Part data of this page collected from the open network resources, so Biochempartner can not guarantee its accuracy.
For product details of different batches, please contact our Customer
Service & Tech Support:orders@biochempartner.com
Website:www.biochempartner.com
Products are for research use only and not for human use. We do not sell to patients.