EST64454 HCl
| CAS No. | 1950569-11-5 | Cat. No. | BCP43797 |
| Name | EST64454 HCl | ||
| Synonyms | EST64454 hydrochloride;EST 64454 HCl;EST-64454 HCl; | ||
| Formula | C18H23ClF2N4O2 | M. Wt | 400.85 |
| Description | EST64454 is a Highly Soluble σ1 Receptor Antagonist Clinical Candidate for Pain Management. EST64454 shows an outstanding aqueous solubility, which together with its high permeability in Caco-2 cells will allow its classification as a BCS class I compound. It also shows high metabolic stability in all species, linked to an adequate pharmacokinetic profile in rodents, and antinociceptive properties in the capsaicin and partial sciatic nerve ligation models in mice. | ||
| Pathways | GPCR/G Protein | ||
| Targets | Sigma Receptor | ||
Structure
Part data of this page collected from the open network resources, so Biochempartner can not guarantee its accuracy.
For product details of different batches, please contact our Customer
- Service & Tech Support:orders@biochempartner.com
- Website:www.biochempartner.com
Products are for research use only and not for human use. We do not sell to patients.