Omarigliptin
| CAS No. | 1226781-44-7 | Cat. No. | BCP08054 |
| Name | Omarigliptin | ||
| Synonyms | MK3102; MK 3102:MK-3102; | ||
| Formula | C17H20F2N4O3S | M. Wt | 398.43 |
| Description | Omarigliptin (MK-3102) is a competitive, reversible inhibitor of DPP-4 (IC50 = 1.6 nM, Ki = 0.8 nM). It is highly selective over all proteases tested (IC50 > 67 μM), including QPP, FAP, PEP, DPP8, and DPP9 and has weak ion channel activity (IC50 > 30 μM at IKr, Caγ1.2, and Naγ1.5). | ||
| Pathways | Protease/Metabolic Enzyme | ||
| Targets | DPP | ||
Structure
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