CNV-1014802
| CAS No. | 934240-30-9 | Cat. No. | BCP07060 |
| Name | CNV-1014802 | ||
| Synonyms | GSK-1014802;GSK 1014802;GSK1014802;CNV1014802;CNV 1014802;Raxatrigine; | ||
| Formula | C18H19FN2O2 | M. Wt | 314.35 |
| Description | Raxatrigine, also known as GSK1014802 and CNV-1014802, is a sodium channel antagonist that is currently in phase II studies in bipolar depression. CNV1014802 is a peripherally and centrally acting agent that inhibits sodium channels in a state-dependent fashion. CNV1014802 shows selectivity for the Nav1.7 subtype over the other subtypes tested (Nav1.1, Nav1.2, Nav1.3, Nav1.5, Nav1.6 and TTX-R), for both the resting and depolarized states. | ||
| Pathways | Ion Channel/Membrane Transporter | ||
| Targets | Sodium Channel | ||
Structure
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