Carbazeran
| CAS No. | 70724-25-3 | Cat. No. | BCP06512 |
| Name | Carbazeran | ||
| Synonyms | UK 31557;UK-31557;UK31557; | ||
| Formula | C18H24N4O4 | M. Wt | 360.412 |
| Description | Carbazeran is an Aldehyde oxidase (AO) substrate and potent phosphodiesterase PDE-II and PDE-III inhibitor that produces concentration-dependent positive inotropic responses. Carbazeran shows chronotropic and inotropic effect in vivo (EC50 = 100 μM, ionotropic effects, independent of adrenergic mechanisms). It potently inhibits cAMP hydrolysis. In humans, the compound is almost completely cleared via 4-hydroxylation to the phthalazinone metabolite by AO. | ||
| Pathways | Protease/Metabolic Enzyme | ||
| Targets | Phosphodiesterase/PDE | ||
Structure
Part data of this page collected from the open network resources, so Biochempartner can not guarantee its accuracy.
For product details of different batches, please contact our Customer
- Service & Tech Support:orders@biochempartner.com
- Website:www.biochempartner.com
Products are for research use only and not for human use. We do not sell to patients.