G007-LK
| CAS No. | 1380672-07-0 | Cat. No. | BCP11079 |
| Name | G007-LK | ||
| Synonyms | G007LK; G007 LK; | ||
| Formula | C25H16ClN7O3S | M. Wt | 529.96 |
| Description | G007-LK is a potent, "rule of 5" compliant and a metabolically stable TNKS1/2 inhibitor. G007-LK displayed high selectivity toward tankyrases 1 and 2 with biochemical IC50 values of 46 nM and 25 nM, respectively, and a cellular IC50 value of 50 nM combined with an excellent pharmacokinetic profile in mice. G007-LK was first discovered by Dr. Stefan Krauss's team. | ||
| Pathways | Cell Cycle/DNA Damage Epigenetics | ||
| Targets | PARP | ||
Structure
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