Meptazinol hydrochloride

  • Chemical Properties
CAS No. 59263-76-2 Cat. No. BCP12143
Name Meptazinol hydrochloride
Synonyms Meptazinol HCl; IL 22811 HCl; IL-22811 HCl; IL22811 HCl; WY 22811 HCl; WY-22811 HCl; WY22811 HCl;
Formula C15H23NO.HCl M. Wt 269.81
  • Biological Activity
Description Meptazinol Hcl(WY-22811 Hcl) is a unique centrally active opioid analgesic.Meptazinol is an opioid analgesic developed by Wyeth in the 1970s. Indications for use in moderate to severe pain, most commonly used to treat pain in obstetrics (childbirth). Meptazinol is a 3-phenylazpane derivative, whereas the other phenazepanes like ethoheptazine and proheptazine are 4-phenylazepanes. A partial µ-opioid receptor agonist, its mixed agonist/antagonist activity affords it a lower risk of dependence and abuse than full µ agonists like morphine. Meptazinol exhibits not only a short onset of action, but also a shorter duration of action relative to other opioids such as morphine, pentazocine, or buprenorphine.
Pathways Neuro Signaling Pathway Hormone Pathay GPCR/G Protein 
Targets Opioid Receptor 

Structure

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