氢溴酸替格列汀
CAS号 | 906093-29-6 | 货号 | BCP12262 |
中文名 | 氢溴酸替格列汀 | ||
英文名 | Teneligliptin hydrobromide | ||
中文别名 | |||
英文别名 | Teneligliptin HBr;MP-513 hydrobromide;MP513 hydrobromide; | ||
分子式 | 2(C22H30N6OS).5(HBr) | 分子量 | 1257.72 |
生物活性 | Teneligliptin hydrobromide is a potent chemotype prolylthiazolidine-based DPP-4 inhibitor, which competitively inhibits human plasma, rat plasma, and human recombinant DPP-4 in vitro, with IC50s of approximately 1 nM.Teneligliptin is a pharmaceutical drug for the treatment of type 2 diabetes mellitus. It belongs to the class of anti-diabetic drugs known as dipeptidyl peptidase-4 inhibitors or "gliptins". It is approved for use in Japan. | ||
信号通路 | Protease/Metabolic Enzyme | ||
靶 点 | DPP |
结构式

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