Tirolisant
CAS No. | 362665-56-3 | Cat. No. | BCP13114 |
Name | Tirolisant | ||
Synonyms | BF2649; BF-2649; BF 2649; Pitolisant; | ||
Formula | C17H26ClNO | M. Wt | 295.85 |
Description | Pitolisant, also known as Tiprolisant, BF2649, is a histamine receptor inverse agonist/antagonist selective for the H3 subtype. It has stimulant and nootropic effects in animal studies, and may have several medical applications, having been researched for the treatment of narcolepsy, for which it has been granted orphan drug status in the EU and US. It is currently in clinical trials for schizophrenia and Parkinson's disease. Pitolisant was the first clinically used H3 receptor inverse agonist. | ||
Pathways | Neuro Signaling Pathway GPCR/G Protein | ||
Targets | Histamine Receptor |
Structure
Part data of this page collected from the open network resources, so Biochempartner can not guarantee its accuracy.
For product details of different batches, please contact our Customer
- Service & Tech Support:orders@biochempartner.com
- Website:www.biochempartner.com
Products are for research use only and not for human use. We do not sell to patients.