Cebranopadol hemicitrate

  • Chemical Properties
CAS No. 863513-92-2 Cat. No. BCP18808
Name Cebranopadol hemicitrate
Synonyms GRT-6005 hemicitrate; GRT 6005 hemicitrate; GRT6005 hemicitrate;
Formula C54H62F2N4O9 M. Wt 949.09
  • Biological Activity
Description Cebranopadol, also known as GRT-6005, is a Opioid Receptor Agonist with agonistic activity at nociceptin/orphanin FQ and opioid receptors. Cebranopadol displays analgesic, antiallodynic and antihyperalgesic properties in several rat models of acute nociceptive, inflammatory, cancer and neuropathic pain. In contrast to classical opioids, it has a higher analgesic potency in models of neuropathic pain than in acute nociceptive pain. Even at higher analgesic doses, cebranopadol does not induce motor coordination deficits or respiratory depression in rats.
Pathways Neuro Signaling Pathway Hormone Pathay GPCR/G Protein 
Targets Opioid Receptor 

Structure

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