Rapastinel acetate
CAS No. | 491872-39-0 | Cat. No. | BCP24900 |
Name | Rapastinel acetate | ||
Synonyms | GLYX-13; GLYX 13; GLYX13; BV-102; BV102; BV 102; TPPT-amide; | ||
Formula | C20H35N5O8 | M. Wt | 473.52 |
Description | Rapastinel is a novel antidepressant drug approved as an adjunctive therapy for the treatment of treatment-resistant major depressive disorder. It is a centrally active, intravenously administered (non-orally active) amidated tetrapeptide (Thr-Pro-Pro-Thr-NH2) that acts as a selective, weak partial agonist (mixed antagonist/agonist) of an allosteric site at the glycine site of the NMDA receptor complex (Emax ≈ 25%). | ||
Related Products | 1435786-04-1(Rapastinel Trifluoroacetate) | ||
Pathways | Neuro Signaling Pathway GPCR/G Protein | ||
Targets | mGluR |
Structure
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