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GDC-0032 Chemical Structure

GDC-0032

Data Sheet For research use only. Not for human use.
Cat. No. ：BCP09253CAS No. ：1282512-48-4Purity：98%
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  • Chemical Properties&Biological Activity
CAS No. 1282512-48-4 Cat. No. BCP09253
Name GDC-0032
Synonyms Taselisib; RG7604;RG-7604; GDC0032; GDC 0032;
SMILES
Chemical Name
Formula C24H28N8O2 M. Wt 460.53
Purity 98% Storage Store at 4-8°C
Description GDC-0032 is an orally bioavailable, potent and selective inhibitor of Class I PI3Kα, δ and γ isoforms, with 30 fold less inhibition of the PI3K β isoform relative to the PI3Kα isoform. GDC-0032 inhibits MCF7-neo/HER2 cells proliferation with IC50 of 2.5 nM. The combination of GDC-0032 with tamoxifen enhances the efficacy of tamoxifen in vivo (102%TGI for GDC-0032). GDC-0032 is currently in a phase I clinical trial.
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H-NMR
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