CCT251921
Data Sheet
For research use only. Not for human use.
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| CAS No. | 1607837-31-9 | Cat. No. | BCP19641 |
| Name | CCT251921 | ||
| Synonyms | CCT-251921;CCT 251921; | ||
| SMILES | |||
| Chemical Name | |||
| Formula | C21H23ClN6O | M. Wt | 410.9 |
| Purity | 98% | Storage | Store at 4-8°C |
| Description | CCT251921 is a potent, selective, and orally bioavailable small-molecule modulators of the mediator complex-associated kinases CDK8 and CDK19. (IC50 data: CDK8:=2.3 nM; CDK19 = 2.6 nM). CCT251921 showed the optimal compromise of in vitro biochemical, pharmacokinetic, and physicochemical properties and is suitable for progression to animal models of cancer. The Mediator complex-associated cyclin-dependent kinase CDK8 has been implicated in human disease, particularly in colorectal cancer where it has been reported as a putative oncogene. | ||
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