MSC2530818
Data Sheet
For research use only. Not for human use.
Get Quotation Now* Required Fields.
Please complete the form below and you will get the price list in 1 minute.
* Required Fields.
Please complete the form below and we will contact you shortly.
* Required Fields.
Please complete the form below and we will contact you shortly.
| CAS No. | 1883423-59-3 | Cat. No. | BCP20854 |
| Name | MSC2530818 | ||
| Synonyms | MSC-2530818;MSC 2530818; | ||
| SMILES | O=C(N1[C@](C2=CC=C(Cl)C=C2)CCC1)C3=CN=C(NN=C4C)C4=C3 | ||
| Chemical Name | |||
| Formula | C18H17ClN4O | M. Wt | 340.81 |
| Purity | 98% | Storage | Store at 4-8°C |
| Description | MSC2530818 is a Potent, Selective, and Orally Bioavailable CDK8 Inhibitor with CDK8 IC50 = 2.6 nM; Human PK prediction: Cl ~ 0.14 L/H/Kg; t1/2 ~ 2.4h; F > 75%. MSC2530818 displays excellent kinase selectivity, biochemical and cellular potency, microsomal stability, and is orally bioavailable. MSC2530818 demonstrates suitable potency and selectivity to progress into preclinical in vivo efficacy and safety studies. | ||
Recommend Products
More >
-
-
Inixaciclib
Cat. No.：BCP49218
No.：2370913-42-9
Product Details -
FMF-04-159-2
Cat. No.：BCP48874
No.：2364489-81-4
Product Details -
-
GSK-3/CDK5/CDK2-IN-1
Cat. No.：BCP48519
No.：395074-72-3
Product Details -
LY3143921 hydrate
Cat. No.：BCP48020
No.：1627696-53-0
Product Details -
LY3143921
Cat. No.：BCP48019
No.：1627696-52-9
Product Details -
-
Cdk2/9 Inhibitor
Cat. No.：BCP46934
No.：507487-89-0
Product Details -
Aminopurvalanol A
Cat. No.：BCP46783
No.：220792-57-4
Product Details -
-
-
-
CDK12-IN-2
Cat. No.：BCP46385
No.：2244987-03-7
Product Details -
CDK4/6-IN-6
Cat. No.：BCP46270
No.：2380321-51-5
Product Details -
CDK5-IN-3
Cat. No.：BCP46220
No.：2639542-32-6
Product Details -
KB-0742 hydrochloride
Cat. No.：BCP36919
No.：2416874-75-2
Product Details -
(-)-BAY-1251152
Cat. No.：BCP33291
No.：1610358-59-2
Product Details -
Fascaplysin
Cat. No.：BCP24646
No.：114719-57-2
Product Details -
Aloisine A
Cat. No.：BCP26893
No.：496864-16-5
Product Details
Tags:MSC2530818 supplier,MSC2530818 purchase,MSC2530818 manufacturer,MSC2530818 distributor,MSC2530818 cost,MSC2530818 buy,MSC2530818 for sale