AZD7545
Data Sheet
For research use only. Not for human use.
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| CAS No. | 252017-04-2 | Cat. No. | BCP07524 |
| Name | AZD7545 | ||
| Synonyms | AZD 7545; AZ-7545; | ||
| SMILES | |||
| Chemical Name | |||
| Formula | C19H18ClF3N2O5S | M. Wt | 478.87 |
| Purity | 98% | Storage | Store at 4-8°C |
| Description | AZD7545 is a novel, selective small-molecule inhibitor of PDHK2 (PDH kinase2) with an IC50 of 36.8 nM and 6.4 nM for PDHK1 and PDHK2 respectively. IC50 Value: 36.8 nM (PDHK1); 6.4 nM (PDHK2) [1] Target: PDHK in vitro: The IC50 values for inhibition of PDHK2 and PDHK1 by AZD7545 were 6.4 ± 2.2 nM (n = 6) and 36.8 ± 18 nM (n = 3) respectively. Other compounds in this series inhibited both PDHK1 and PDHK2 and a consistent trend of reduced potency (5-15-fold) towards PDHK1, as compared with PDHK2, | ||
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