Cas No.Product NameDescription
81065-76-1EUK-134EUK 134 is a synthetic manganese-porphyrin complexe which has been documented to act as a scavenger for oxidative species such as hydrogen peroxide, peroxynitrite and superoxide.
150322-43-3PrasugrelPrasugrel is a member of the thienopyridine class of ADP receptor inhibitors.
957118-49-9MK 3207MK-3207 is a potent and orally bioavailable CGRP receptor antagonist. In common with other CGRP receptor antagonists, MK-3207 displays lower affinity for human CGRP receptors from other species, including canine and rodent.
74711-43-6ZaltoprofenZaltoprofen is an inhibitor of Cox-1 and Cox-2 for treatment of arthritis.
501925-31-1PNU120596PNU-120596 is a positive allosteric modulator of α7 nAChR with EC50 of 216 nM.
4460-86-0 AcroleinAsaraldehyde is a natural COX-2 inhibitor, exhibiting 17-fold selectivity over COX-1.
15307-79-6Diclofenac sodiumDiclofenac Sodium is a non-selective COX inhibitor with IC50 of 60 and 220 nM for ovine COX-1 and -2, respectively.
74103-07-4Ketorolac Ketorolac (Ketorolac tromethamine) is a non-selective COX inhibitor of COX-1 and COX-2 with IC50 of 1.23 μM and 3.50 μM, respectively.
85375-15-1SKF 89976A HClSKF 89976A is a GABA transporter type 1 inhibitor with IC50 of 0.13, 550, 944 and 7210 μM for hGABA T-1, rGABa T-2, hGABA T-3 and hBGT-1 respectively. SKF-89976A is selective for GABA T-1. This compound inhibits transport current competitively (Ki = 7 μM) and transmitter-gated current non-competitively.
300-08-3 Arecoline hydrobromideArecoline Hydrobromide is a muscarinic acetylcholine receptor agonist.
139404-48-1Tiotropium Bromide hydrateTiotropium Bromide hydrate is an anticholinergic and bronchodilator and a muscarinic receptor antagonist.
136310-93-5Tiotropium BromideTiotropium Bromide is a muscarinic acetylcholine receptor (mAChR M) antagonist that blocks the binding of the acetylcholine ligand and subsequent opening of the ligand-gated ion channel.
124937-52-6Tolterodine tartrateTolterodine tartrate (Detrol LA) is a tartrate salt of tolterodine that is a competitive muscarinic receptor antagonist. Tolterodine tartrate (Detrol LA) is indicated for the treatment of overactive bladder with symptoms of urge urinary incontinence, urgency and frequency.
1104-22-9Meclizine HClMeclizine is a histamine H1 receptor antagonist used to treat nausea and motion sickness, has anti-histamine, anti-muscarinic and anti-oxidative phosphorylation properties, also an agonist ligand for mCAR (constitutive androstane receptor) and an inverse agonist for hCAR.
119302-91-9Rocuronium bromideRocuronium is an aminosteroid non-depolarizing neuromuscular blocker or muscle relaxant used in modern anaesthesia, to facilitate endotracheal intubation and to provide skeletal musclerelaxation during surgery or mechanical ventilation.
1246086-78-1VU 0364439Positive allosteric modulator (PAM) of mGlu4 receptors (EC50 = 19.8 nM in vitro for human mGlu4).
50700-72-6Vecuronium bromideVecuronium (bromide) is a muscle relaxant in the category of non-depolarizing blocking agents.
1953-04-4Galanthamine hydrobromideGalanthamine is an AChE inhibitor with IC50 of 0.35 μM, exhibits 50-fold selectivity against butyryl-cholinesterase.

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Cell Cycle/Checkpoint
Angiogenesis/Tyrosine Kinase
Apoptosis Pathway
Aurora/Ksp Pathway
MAPK Pathway
Hormone Pathay
Proteases/HSP90/HSP70 Pathway
Wnt/Hedgehog/Notch Pathway
Jak/Stat Pathway
Ca/cAMP/Lipid Signaling Pathway
Neuro Signaling Pathway
TGF-beta/Smad Signaling Pathway
GPCR Pathway
Ion channel Pathway
Cytochrome P450 Pathway
Others Pathway