Relacorilant
| CAS No. | 1496510-51-0 | Cat. No. | BCP30640 |
| Name | Relacorilant | ||
| Synonyms | CORT125134; CORT-125134; CORT 125134; | ||
| Formula | C27H22F4N6O3S | M. Wt | 586.56 |
| Description | Relacorilant is a potent, selective and orally bioavailable glucocorticoid receptor antagonist, with a Ki of 7.2 nM in HepG2 TAT assay, and also shows Kis of 12, 81.2, 210 nM for rat, human and monkey glucocorticoid receptor in cell-based assay, respectively; Relacorilant has entered phase 2 clinical study in patients with Cushing’s syndrome. | ||
| Pathways | GPCR/G Protein | ||
| Targets | Glucocorticoid Receptor | ||
Structure
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