TP-064
| CAS No. | 2080306-20-1 | Cat. No. | BCP43164 |
| Name | TP-064 | ||
| Synonyms | TP 064; TP064; | ||
| Formula | C28H34N4O2 | M. Wt | 458.6 |
| Description | TP-064 is a potent and selective PRMT4 inhibitor. The in vitro activity of TP-064 includes inhibition of PRMT4 with IC50 < 10nM for methylation of H3 (1-25) and greater than 100-fold selectivity over other histone methyltransferases and non-epigenetic targets. In cellular assays, TP-064 inhibits the methylation of MED12 with IC50 = 43 nM. | ||
| Pathways | Epigenetics | ||
| Targets | Histone Methyltransferase | ||
Structure
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