RVX297
| CAS号 | 1044871-04-6 | 货号 | BCP43937 |
| 中文名 | RVX297 | ||
| 英文名 | RVX297 | ||
| 中文别名 | |||
| 英文别名 | RVX 297; RVX-297; | ||
| 分子式 | C24H29N3O4 | 分子量 | 423.5 |
| 生物活性 | RVX-297 is a BD2 selective inhibitor of BET bromodomains. RVX-297 is structurally related to the clinical compound RVX-208, currently undergoing phase III clinical trials for the treatment of cardiovascular diseases, but is distinctly different in its biological and pharmacokinetic profiles. RVX-297 preferentially binds to the BD2 domains of the BET bromodomain and Extra Terminal (BET) family of protein. Selective inhibition of either BD1 or BD2 can have significant implications on differential gene expression, which possibly can be further linked to the specific disease indication. | ||
| 信号通路 | Epigenetics | ||
| 靶 点 | Epigenetic Reader Domain | ||
结构式
本页面部分数据来自于公开的网络资源,所以瀚香生物不能保证其准确性。
不同批次的产品详情请咨询我们的客服：
- 全国免费电话：400-099-8200
- 在线客服:
瀚香生物（Biochempartner) 的所有产品和服务仅用于科学研究，禁止用于人体和治疗！