PF429242

  • Chemical Properties
CAS No. 947303-87-9 Cat. No. BCP03764
Name PF429242
Synonyms PF 429242;PF-429242;
Formula C25H35N3O2 M. Wt 409.56
  • Biological Activity
Description Reversible, competitive inhibitor of sterol regulatory element-binding protein (SREBP) site 1 protease (IC50 = 0.175 μM). Selective for site 1 protease against a panel of serine proteases. Inhibits rate of cholesterol synthesis in CHO cells (IC50 = 0.53 μM). Also displays antiviral activity. Cell permeable.
Related Products 2248666-66-0(PF429242 dihydrochloride)
Pathways GPCR/G Protein 
Targets S1P Receptor 

Structure

Part data of this page collected from the open network resources, so Biochempartner can not guarantee its accuracy.
For product details of different batches, please contact our Customer
Service & Tech Support:orders@biochempartner.com
Website:www.biochempartner.com
Products are for research use only and not for human use. We do not sell to patients.