盐酸瑞伐拉赞
| CAS号 | 178307-42-1 | 货号 | BCP09645 |
| 中文名 | 盐酸瑞伐拉赞 | ||
| 英文名 | Revaprazan Hydrochloride | ||
| 中文别名 | 盐酸洛氟普啶; | ||
| 英文别名 | Revaprazan HCl;SB 641257 Hydrochloride;SB 641257A; YH 1885; YH-1885; YH1885; | ||
| 分子式 | C22H24ClFN4 | 分子量 | 398.9 |
| 生物活性 | Revaprazan Hydrochloride is the hydrochloride salt form of a lipophilic, weak base with potassium-competitive acid blocking (P-CAB) activity. Revaprazan concentrates highly in the gastric parietal cell canaliculus and on entering this acidic environment is instantly protonated and binds competitively and reversibly to the potassium binding site of the proton pump hydrogen-potassium adenosine triphosphatase (H+/K+ ATPase), thereby inhibiting the pump's activity and the parietal cell secretion of H+ ions into the gastric lumen, the final step in gastric acid production. | ||
| 信号通路 | Ion Channel/Membrane Transporter | ||
| 靶 点 | Potassium Channel | ||
结构式
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