EMPA
| CAS No. | 680590-49-2 | Cat. No. | BCP23952 |
| Name | EMPA | ||
| Synonyms | 7MA; | ||
| Formula | C23H26N4O4S | M. Wt | 454.54 |
| Description | EMPA is a highly potent, selective OX2 receptor antagonist (IC50 values are 2.3 nM and 1900 nM for OX2 and OX1 respectively). Displays negligible or no inhibition of a panel of 80 receptors. Blocks orexin-B- and orexin-A-invoked calcium mobilization in hOX2-expressing CHO cells (IC50 values are 7.9 nM and 8.8 nM respectively); reverses orexin-B-induced hyperlocomotion in mice. Brain penetrant. | ||
| Pathways | GPCR/G Protein | ||
| Targets | OX Receptor | ||
Structure
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