Tebanicline benzoate
| CAS号 | 209326-18-1 | 货号 | BCP25230 |
| 中文名 | Tebanicline benzoate | ||
| 英文名 | Tebanicline benzoate | ||
| 中文别名 | |||
| 英文别名 | Ebanicline benzoate;ABT594 benzoate; | ||
| 分子式 | C16H17ClN2O3 | 分子量 | 320.77 |
| 生物活性 | Tebanicline acts as a partial agonist at neuronal nicotinic acetylcholine receptors, binding to both the α3β4 and the α4β2 subtypes. Tebanicline is an effective synthetic nicotinic (non-opioid) analgesic drug developed by Abbott. It was developed as a less toxic analog of the potent poison dart frog-derived compound epibatidine, which is some 200x stronger than morphine as an analgesic but produces extremely dangerous toxic side effects. Like epibatidine, Tebanicline showed potent analgesic activity against neuropathic pain in both animal and human trials, but with far less toxicity than its parent compound. | ||
| 上下游产品 | 198283-74-8（Tebanicline tosylate） 209326-19-2（Tebanicline dihydrochloride） 203564-54-9（Tebanicline HCl） 198283-73-7（Tebanicline） | ||
| 信号通路 | Ion Channel/Membrane Transporter Neuro Signaling Pathway | ||
| 靶 点 | nAChR | ||
结构式
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