Rolapitant
Data Sheet
For research use only. Not for human use.
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| CAS No. | 552292-08-7 | Cat. No. | BCP09609 |
| Name | Rolapitant | ||
| Synonyms | (5S,8S)-8-[[(1R)-1-[3,5-bis(trifluoromethyl)phenyl]ethoxy]methyl]-8-phenyl-1,9-diazaspiro[4.5]decan-2-one; | ||
| SMILES | |||
| Chemical Name | |||
| Formula | C25H26F6N2O2 | M. Wt | 500.48 |
| Purity | 98% | Storage | Store at 4-8°C |
| Description | . In vitro studies indicate that rolapitant has a high affinity for the human NK1 receptor of 0.66 nM and high selectivity over the human NK2 and NK3 subtypes of >1000-fold. Rolapitant is a functionally competitive antagonist, as measured by calcium efflux, with a calculated Kb of 0.17 nM. | ||
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