Elacestrant New

Data Sheet For research use only. Not for human use.

Cat. No. ：BCP39541CAS No. ：722533-56-4Purity：98%

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CAS No.	722533-56-4	Cat. No.	BCP39541
Name	Elacestrant
Synonyms	RAD1901; RAD-1901; RAD 1901;
SMILES	CCNCCC1=CC=C(C=C1)CN(CC)C2=C(C=CC(=C2)OC)C3CCC4=C(C3)C=CC(=C4)O
Chemical Name
Formula	C30H38N2O2	M. Wt	458.63
Purity	98%	Storage	Store at 4-8°C
Description	Elacestrant is an orally available, selective estrogen receptor degrader (SERD) and selective estrogen receptor modulator (SERM), with potential antineoplastic and estrogen-like activities. Upon oral administration of higher doses of RAD1901, this agent acts as a SERD, which binds to the estrogen receptor (ER) and induces a conformational change that results in the degradation of the receptor. This may inhibit the growth and survival of ER-expressing cancer cells. At lower doses of this agent, RAD1901 acts as a SERM and has estrogen-like effects in certain tissues, which can both reduce hot flashes and protect against bone loss. In addition, RAD1901 is able to cross the blood-brain barrier (BBB).