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Paltusotine Chemical Structure

Paltusotine

Data Sheet For research use only. Not for human use.
Cat. No. :BCP47002CAS No. :2172870-89-0Purity:98%
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  • Chemical Properties&Biological Activity
CAS No. 2172870-89-0 Cat. No. BCP47002
Name Paltusotine
Synonyms CRN00808; CRN-00808; CRN 00808;
SMILES C1CN(CCC1N)C2=C3C=C(C=CC3=NC=C2C4=CC(=CC(=C4)F)F)C5=CC=CC(=C5O)C#N
Chemical Name
Formula C27H22F2N4O M. Wt 456.49
Purity 98% Storage Store at 4-8°C
Description Paltusotine is an orally bioavailable, nonpeptide somatostatin receptor type 2 (SST2; SSTR2) agonist, with potential growth hormone (GH) secretion-inhibiting and antineoplastic activities. Upon oral administration, paltusotine targets, binds to and activates SSTR2, which leads to an inhibition in the secretion of human growth hormone (hGH) in the pituitary gland and results in decreased production of insulin-like growth factor (IGF-1). This may inhibit IGF-1-mediated cell signaling pathways, and lead to apoptosis. SSTR2 is overexpressed by some neuroendocrine tumor cells, and GH is over-produced in the pituitary gland in acromegaly.
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