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Rolapitant Chemical Structure

Rolapitant

Data Sheet For research use only. Not for human use.
Cat. No. :BCP09609CAS No. :552292-08-7Purity:98%
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  • Chemical Properties&Biological Activity
CAS No. 552292-08-7 Cat. No. BCP09609
Name Rolapitant
Synonyms (5S,8S)-8-[[(1R)-1-[3,5-bis(trifluoromethyl)phenyl]ethoxy]methyl]-8-phenyl-1,9-diazaspiro[4.5]decan-2-one;
SMILES
Chemical Name
Formula C25H26F6N2O2 M. Wt 500.48
Purity 98% Storage Store at 4-8°C
Description . In vitro studies indicate that rolapitant has a high affinity for the human NK1 receptor of 0.66 nM and high selectivity over the human NK2 and NK3 subtypes of >1000-fold. Rolapitant is a functionally competitive antagonist, as measured by calcium efflux, with a calculated Kb of 0.17 nM.
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