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CAS号 | 372523-75-6 | 货号 | BCP20353 |
中文名 | TCS-OX2-29 | ||
英文名 | TCS-OX2-29 | ||
中文别名 | |||
英文别名 | |||
SMILES | |||
化学名称 | |||
分子式 | C₂₃H₃₁N₃O₃ | 分子量 | |
纯度 | 98% | 配送 | 惯例下常温包邮 |
产品描述 | Target: OX2 IC 50: 40 nM In vitro:TCS-OX2-29 shows selectivity for ion channels, and transporters (<30% inhibition at 10 μM), which includes G-protein coupled receptors associated with food intake including galanin and neuripeptide Y. [1] TCS-OX2-29 Inhibits orexin A induced IP3 accumulation and ERK1/2 phosphorylation in CHO cells transfected with the OX2 receptor. |
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