所有产品分类
所有产品
信号通路
- Angiogenesis/Protein Tyrosine Kinase
- Apoptosis Pathway
- Cell Cycle/DNA Damage
- Epigenetics
-
GPCR/G Protein
- Urotensin Receptor
- Melatonin Receptor
- Neurotensin Receptor
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- Motilin Receptor
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- Smoothened/Smo
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- Microbiology/Virology
-
Neuro Signaling Pathway
- Imidazoline Receptor
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- FAAH
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- nAChR
- COX
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- mAChR
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-
Protease/Metabolic Enzyme
- COMT
- 11β HSD
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- Xanthine Oxidase
- Pyruvate Kinase
- Mitochondrial Metabolism
- ALDH
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- Serine Protease
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- E1 E2 E3 Enzyme
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- Phosphatase
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- HMGCR
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- Gamma secretase
- RAAS/ACE
- Caspase
- HIV Protease
- Aminopeptidase
- HCV Protease
- HSP
- Tryptophan Hydroxylase/TPH
- Factor Xa
- DPP
- Procollagen C Proteinase
- Integrase
- Phosphodiesterase/PDE
- Phospholipase
- LXR
- Proteasome
- Cytochrome P450
- TGF beta/Smad
- Wnt/Stem Cell
- Others Pathway
研究领域
- Metabolic Disease
- Neurological Disease
- Endocrinology
- Diabetes
- Cardiovascular Disease
- Immunology
- Allergy
- Inflammation
- Infection
- Cancer
天然产物
抗体
多肽
催化剂
杂质对照品
医药中间体
基础原料
Integrase
| 结构式 | 货号 | 产品名称 | CAS号 |
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BCP10394 | BMS-538203 | 543730-41-2 |
BMS-538203 is a highly efficient HIV integrase inhibitor and antiviral agent.
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BCP25703 | 比卡格韦 新 | 1611493-60-7 |
Bictegravir is a novel, potent inhibitor of HIV-1 integrase with an IC50 of 7.5 nM.
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BCP20910 | 比卡格韦纳 新 | 1807988-02-8 |
Bictegravir, also known as GS-9883, is a potent, unboosted, once-Daily HIV-1 Integrase Strand Transfer Inhibitor (INSTI) (IC50 - 1.6 nM) with improved pharmacokinetics and in vitro resistance profile.
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BCP08631 | 卡博特韦 | 1051375-10-0 |
Cabotegravir is a potent HIV integrase inhibitor as an oral lead-in tablet and long-acting injectable for the treatment and prevention of HIV infection. Cabotegravir is an inhibitor of OAT1 (IC50 0.81 μM) and OAT3 (IC50 0.41 μM).
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BCP24687 | 卡博特韦钠盐 | 1051375-13-3 |
Cabotegravir is a potent HIV integrase inhibitor as an oral lead-in tablet and long-acting injectable for the treatment and prevention of HIV infection. Cabotegravir is an inhibitor of OAT1 (IC50 0.81 μM) and OAT3 (IC50 0.41 μM).
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BCP11890 | 度鲁特韦钠盐 新 | 1051375-19-9 |
Dolutegravir sodium salt is a HIV integrase inhibitor(IC50= 2.7 nM), modest activity against raltegravir-resistant signature mutants Y143R, Q148K, N155H, and G140S/Q148H.
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BCP01394 | 雷特格韦 新 | 518048-05-0 |
Raltegravir is a potent integrase (IN) inhibitor, used to treat HIV infection.
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BCP02329 | 度鲁特韦 新 促 | 1051375-16-6 |
Dolutegravir is an integrase inhibitor being developed for the treatment of human immunodeficiency virus (HIV)-1 infection by GlaxoSmithKline (GSK) on behalf of Shionogi-ViiV Healthcare LLC.
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BCP01757 | 雷特格韦钾盐 新 大货 | 871038-72-1 |
Raltegravir Potassium Salt is a potent human immunodeficiency virus (HIV) integrase inhibitor
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BCP01801 | 埃替拉韦 新 | 697761-98-1 |
Elvitegravir is a human immunodeficiency virus integrase inhibitor with EC50 of 0.7, 2.8 and 1.4 for HIV-1 IIIB, HIV-2 EHO and HIV-2 ROD.
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