AR-C155858

参考资料仅供科学研究，不可用于个人用途。

货号：BCP13211CAS号：496791-37-8纯度：98%

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CAS号	496791-37-8	货号	BCP13211
中文名	AR-C155858
英文名	AR-C155858
中文别名
英文别名	AR C155858;ARC155858;
SMILES
化学名称
分子式	C21H27N5O5S	分子量	461.53
纯度	98%	配送	惯例下常温包邮
产品描述	Co-expression of exogenous embigin was without effect on either the expression of MCT1 or its inhibition by AR-C155858. In contrast, expression of active MCT2 at the plasma membrane of oocytes was significantly enhanced by co-expression of exogenous embigin. This additional transport activity was insensitive to inhibition by AR-C155858 unlike that by MCT2 expressed with endogenous basigin that was potently inhibited by AR-C155858. Derived values were 2.3+/-1.4 nM, 1.29+/-0.09 nmol per ml of packed cells and 12.2+/-1.1 s-1 respectively. When expressed in Xenopus laevis oocytes, MCT1 and MCT2 were potently inhibited by AR-C155858, whereas MCT4 was not. Inhibition of MCT1 was shown to be time-dependent, and the compound was also active when microinjected, suggesting that AR-C155858 probably enters the cell before binding to an intracellular site on MCT1 .