Elacestrant 新

参考资料仅供科学研究，不可用于个人用途。

货号：BCP39541CAS号：722533-56-4纯度：98%

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CAS号	722533-56-4	货号	BCP39541
中文名	Elacestrant
英文名	Elacestrant
中文别名
英文别名	RAD1901; RAD-1901; RAD 1901;
SMILES	CCNCCC1=CC=C(C=C1)CN(CC)C2=C(C=CC(=C2)OC)C3CCC4=C(C3)C=CC(=C4)O
化学名称
分子式	C30H38N2O2	分子量	458.63
纯度	98%	配送	惯例下常温包邮
产品描述	Elacestrant is an orally available, selective estrogen receptor degrader (SERD) and selective estrogen receptor modulator (SERM), with potential antineoplastic and estrogen-like activities. Upon oral administration of higher doses of RAD1901, this agent acts as a SERD, which binds to the estrogen receptor (ER) and induces a conformational change that results in the degradation of the receptor. This may inhibit the growth and survival of ER-expressing cancer cells. At lower doses of this agent, RAD1901 acts as a SERM and has estrogen-like effects in certain tissues, which can both reduce hot flashes and protect against bone loss. In addition, RAD1901 is able to cross the blood-brain barrier (BBB).