首页   >  
GPCR/G Protein
  >  
PAR

所有产品分类

所有产品

信号通路

研究领域

天然产物

抗体

多肽

催化剂

杂质对照品

医药中间体

基础原料

PAR

结构式 货号 产品名称 CAS号
SCH 79797 dihydrochloride 结构式
 BCP46793 SCH 79797 dihydrochloride 1216720-69-2
SCH79797 dihydrochloride is a potent, selective non-peptide PAR1 receptor antagonist (IC50 = 70 nM). Inhibits haTRAP-induced- but not γ-thrombin-, ADP- or collagen-induced human platelet aggregation. Also selectively blocks PAR1 agonist- or thrombin-induced increases in cytosolic Ca2+ in vascular smooth muscle cells.
TRAP-6 结构式
 BCP34232 TRAP-6 141136-83-6
TRAP-6, a peptide compound, has been found to be a PAR1 agonist and could also influence the phosphorylation of rapid phosphodiesterase 3A in the positive way.
I-191 结构式
 BCP32684 I-191 1690172-25-8
I-191 is a potent, selective protease-activated receptor 2 (PAR2) antagonist.
SCH 79797 结构式
 BCP21206 SCH 79797 245520-69-8
SCH-79797 is a potent and selective PAR1 antagonist.
AC-264613 结构式
 BCP25509 AC-264613 1051487-82-1
AC-264613 is a novel potent, selective protease-activated receptor PAR2 agonist with potencies ranging from 30-100 nM.
Atopaxar 结构式
 BCP05973 Atopaxar 751475-53-3;943239-67-6
Atopaxar, also known as E5555, is a potent and orally-active PAR-1 inhibitor.
Atopaxar hydrobromide 结构式
 BCP25405 阿托帕沙溴酸 474550-69-1
Atopaxar hydrobromide is a potent, reversible PAR-1 antagonist with IC50 of 19 nM.
AZ 3451 结构式
 BCP29277 AZ 3451 2100284-59-9
AZ 3451 is a potent, and selective PAR2 antagonist with Kd of 13.5 nM; shows excellent selectivity over PAR1 and PAR4 (>50 uM).
ML 161 结构式
 BCP08413 ML 161 423735-93-7
ML-161 is an allosteric inhibitor of PAR1.
FR171113 结构式
 BCP18806 FR171113 173904-50-2
FR 171113 is a protease-activated receptor 1 (PAR1) antagonist displaying significant antiplatelet activity in vitro.
12下一页共 14 条记录 1 / 2 页 
2853530910