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所有产品
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天然产物
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基础原料
TGR5
| 结构式 | 货号 | 产品名称 | CAS号 |
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BCP32623 | SB-756050 新 | 447410-57-3 |
SB-756050 is a selective TGR5 agonist. SB756050 has the potential for type 2 diabetes treatment.
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BCP32736 | SBI-115 新 | 882366-16-7 |
SBI-115 is a TGR5 (GPCR19) antagonist. SBI-115 decreases hepatic cystogenesis with polycystic liver diseases via inhibiting TGR5.
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BCP08750 | TGR5 Receptor Agonist | 1197300-24-5 |
TGR5 Receptor Agonist, a potent TGR5(GPCR19) agonist.
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BCP19638 | BAR502 | 1612191-86-2 |
BAR502 is a dual FXR and GPBAR1 agonist with IC50 values of 2 μM and 0.4 μM, respectively.
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BCP24972 | BAR501 新 | 1632118-69-4 |
BAR501 is a potent, selective GPBAR1 (GPCR19; TGR5) agonist devoid of any FXR agonistic activity, effectively transactivates GPBAR1 in HEK293 cells with EC50 of 1 uM.
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BCP15620 | 去氧胆酸 新 | 83-44-3 |
Deoxycholic acid is specifically responsible for activating the G protein-coupled bile acid receptor TGR5 that stimulates brown adipose tissue (BAT) thermogenic activity.
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