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Sigma Receptor

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Sigma Receptor

结构式 货号 产品名称 CAS号
NE 100 hydrochloride 结构式
 BCP23907 NE 100 hydrochloride 149409-57-4
NE 100 is a potent and selective σ1 receptor antagonist (Ki = 0.86 nM) that displays > 55-fold selectivity over σ2 receptors and > 6000-fold selectivity over D1, D2, 5-HT1A, 5-HT2 and PCP receptors. Exhibits reversible binding (Kd = 1.2 nM) and displays antipsychotic activity in vivo. Orally active.
WQ 1 结构式
 BCP46446 WQ 1 1204401-49-9
WQ 1 is a high affinity and selective σ1 receptor antagonist. It displays σ1/σ2 selectivity ratio of 29512. It Selectively blocks binge eating without a general inhibition of food intake in rats.
Sigma-1 receptor antagonist 2 结构式
 BCP46031 Sigma-1 receptor antagonist 2 1639220-15-7
Sigma-1 receptor antagonist 2 is a potent and selective sigma 1 receptor (σ1 R) antagonist with Kis of 3.88 and 1288 nM for σ1 and σ2 receptor, respectively.
Roluperidone 结构式
 BCP45266 Roluperidone 359625-79-9
Roluperidone is a 5-HT2A and sigma 2 receptor antagonist potentially for the treatment of schizophrenia.
Rimcazole dihydrochloride 结构式
 BCP44459 林卡唑双盐酸盐 75859-03-9
Rimcazole dihydrochloride is a small molecule antagonist of the σ-1 receptor and inhibits tumor cell survival.
EST64454 HCl 结构式
 BCP43797 EST64454 HCl 1950569-11-5
EST64454 is a Highly Soluble σ1 Receptor Antagonist Clinical Candidate for Pain Management.
SR 31747 结构式
 BCP35688 SR 31747 132173-07-0
SR-31747 is a sigma ligand with immunosuppressive and anti-inflammatory properties. SR-31747 blocks cell proliferation by inhibiting sterol isomerase.
BD 1047 结构式
 BCP33959 BD 1047 138356-20-4
BD-1047 is a selective functional antagonist of sigma-1 receptor, shows antipsychotic activity in animal models predictive of efficacy in schizophrenia.
Cutamesine 结构式
 BCP32724 Cutamesine 165377-43-5
Cutamesine (SA4503; AGY-94806) is a selective sigma 1 receptor(σ1R) agonist; high affinity for the sigma 1 receptor subtype labeled by (+)-[3H]pentazocine (IC50= 17.4±1.9 nM); 100-fold less affinity for the sigma 2 receptor.
BD1063 dhydrochloride 结构式
 BCP31637 BD1063 dhydrochloride 206996-13-6
BD1063 dhydrochloride is a potent and selective sigma 1 receptor antagonist.
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